Exemestane

Exemestane research shows potential of estrogen suppression up to 70%

Prevents aromatase enzymes from converting androgen into estrogen

• 90% protein binding with a half life of 27 hours
• Agitate bottle before each administration
• Not for human consumption

Exemestane (also known as Aromasin) is a member of the class of compounds known as aromatase inhibitors. Aromatase is simply an enzyme that synthesizes estrogen. Aromatase inhibitors block the synthesis of estrogen. Exemestane is an irreversible, aromatase inactivator, structurally related to the natural substrate androstenedione. It acts as a false substrate for the aromatase enzyme, and is processed to an intermediate that binds irreversibly to the active site of the enzyme causing its inactivation

Of note: The estrogen suppression rate for Exemestane varies from 35% for estradiol (E2) to 70% for estrone (E1).

CAS Number 107868-30-4

THIS PRODUCT IS NOT INTENDED TO TREAT, CURE OR DIAGNOSE ANY CONDITION OR DISEASE AND IS NOT FOR HUMAN CONSUMPTION